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浜у搧涓庢湇鍔
鐮斿彂涓庡紑鍙
鍏充簬鐮斿彂
鍏徃鎷ユ湁涓€鏀叿鏈夊崥澹€佺澹瓑鍚勫鍘嗗眰娆$粍鎴愮殑200澶氫汉鐨勭爺绌跺垎鏋愬紑鍙戝洟闃燂紝鑰屼笖鍏锋湁涓板瘜鐨勪粠涓氱粡楠屻€侟/p>
涓轰簡纭繚鐮斿彂鐨勬晥鐜囧拰璐ㄩ噺锛屽叕鍙告垚绔嬩簡涓€涓敱闄㈠+銆佹暀鎺堛€佸崥澹拰涓撳缁勬垚鐨勯【闂洟闃燂紝涓哄叕鍙哥殑鐮旂┒寮€鍙戝嚭璋嬪垝绛栥€侟/p>
鍦ㄨ嚜涓荤爺鍙戠殑鍚屾椂锛屽叕鍙歌繕涓庡浗鍐呭鐭ュ悕鐨勯櫌鎵€寮€灞曚簡绱у瘑鐨勬í鍚戝悎浣滐紝鐩墠宸蹭笌涓浗鍖诲绉戝闄€侀儜宸炲ぇ瀛︺€佹禉姹熷ぇ瀛︺€佷腑绉戦櫌涓婃捣鏈夋満鍖栧鐮旂┒鎵€銆佸寳浜寲宸ュぇ瀛︾瓑鍗曚綅杩涜鍚堜綔锛屽厖鍒嗗彂鎸ヤ骇銆佸銆佺爺浜掑姩浼樺娍锛屾彁鍗囩爺鍙戞晥鐜囥€傜揣瀵嗙殑鍚堜綔涓嶄粎鏈夋晥鐨勫姞寮鸿祫婧愭暣鍚堬紝鍚屾椂涔熷ぇ澶х殑鎻愰珮浜嗗叕鍙告妧鏈垱鏂扮殑閫熷害鍜屽姏搴︼紝涓哄叕鍙哥殑鍙戝睍鎻愪緵浜嗗己鏈夊姏鐨勬妧鏈敮鎾戙€侟/p>
鍏徃鐮斿彂宸ヤ綔浠ユ湇鍔$敓浜у拰甯傚満涓烘牳蹇冿紝涓昏浠ュ伐鑹虹爺鍙戜负涓汇€侟/p>
鎸夌収GMP鐨勮姹傦紝鍦ㄨ瀹氱殑鏃堕棿鍐咃紝灏嗙爺鍙戞垚鏋滆繀閫熻浆鍖栦负宸ヤ笟鐢熶骇锛屾弧瓒冲鎴风殑闇€姹傛槸鎴戜滑鐨勭壒闀裤€侟/p>
鐮斿彂鑳藉姏
鍙嶅簲娓╁害锛?100°C to 400°C
鍙嶅簲鍘嬪姏锛氫粠甯稿帇鍒 10MPa;
鐩墠鐢熶骇涓婃搮闀跨殑鐢熶骇鎶€鏈富瑕佹湁锛欬br />
Chiral technology
Grignard reaction
BuLi reaction
Catalytic reduction
Oxidation reaction
Halogenation reaction
Friedel Crafts reaction
Alkylation reaction
Esterification reaction
Hydrolysis reaction
Phosgene substitution reaction
Nitration reaction
Diazotization reaction
Cross-coupling reaction
Borane reaction
閰跺伐绋
鎴戜滑鐨勯叾宸ョ▼鍥㈤槦涓撴敞浜庝互鏁版嵁鍜屾ā鍨嬮┍鍔ㄧ殑鐢熺墿鍌寲宸ヨ壓寮€鍙戯紝閲囩敤鏅鸿兘閰跺彂鐜版祦绋嬶紝灏嗙敓鐗╀俊鎭銆佺墿鐞嗘ā鎷熶笌鏈哄櫒瀛︿範鏈夋満缁撳悎銆傛垜浠槸E.coli銆丳.pastoris銆丼.cerevisiae鍙夿acillus绛夎〃杈剧郴缁熺殑涓撲笟鐮斿彂涓撳锛屽苟鎷ユ湁鑷富鐮斿彂鐨勯叾搴擄紝鍏朵腑鏀跺綍浜嗚秴杩?000绉嶉叾锛屾兜鐩栬嵂鐗╁悎鎴愭墍闇€鐨勬墍鏈夊叧閿被鍒€傛垜浠殑鍙戦叺鑳藉姏瑕嗙洊浠?鍗囧埌20绔嬫柟绫筹紙姣忓懆鏈€楂樺彲杈?0,000鍗囷級锛屽苟鑳藉疄鐜颁粠鎽囩摱鍩瑰吇鍒版壒閲忕敓浜х殑蹇€熷钩琛屽彂閰靛紑鍙戯紝鍛ㄦ湡浠呴渶鏁板懆銆傜洰鍓嶏紝鎴戜滑宸叉垚鍔熷疄鐜颁簡澶氶」搴旂敤妗堜緥锛屼緥濡侻NR-01銆侀叜杩樺師閰?閱囪劚姘㈤叾绛変骇鍝併€侟/p>
澶氳偨
鎴戜滑澶氳偨鍥㈤槦鐨勭獊鍑轰紭鍔垮湪浜庡崜瓒婄殑澶氳偨鍚堟垚銆佺函鍖栦笌淇グ鎶€鏈兘鍔涳紙鍖呮嫭鍥虹浉鑲藉悎鎴愭硶銆佹恫鐩歌偨鍚堟垚娉曪紝浠ュ強缁撳悎鍥虹浉涓庢恫鐩哥殑娣峰悎鏂规硶锛涘悓鏃舵帉鎻″鑲芥瀯寤烘ā鍧楀悎鎴愭妧鏈瓑锛夈€傛澶栵紝鍥㈤槦杩樼簿閫氬绉嶄繚鎶ょ瓥鐣ワ紙濡侳moc銆乼-Boc銆丆bz绛夛級鍙婂叏闈㈢殑澶氳偨淇グ鎶€鏈綋绯伙紙娑电洊姘ㄥ熀閰镐晶閾句慨楗般€佹湯绔慨楗般€佺幆鍖栦慨楗般€丳EG鍖栦慨楗般€佽崸鍏夋爣璁颁慨楗般€佺敓鐗╃礌鍖栦慨楗般€佺硸鍩哄寲淇グ锛屼互鍙婂悓浣嶇礌鏍囪淇グ绛夊绉嶅墠娌挎妧鏈級銆侟br>鎴戜滑鎻愪緵鍏ㄦ柟浣嶇殑澶氳偨浜т笟鍖栨湇鍔★細鍖呮嫭澶氳偨鏋勫缓妯″潡銆佸鑲藉師鏂欒嵂寮€鍙戜笌鐢熶骇锛屼互鍙婂鑲紺DMO鏈嶅姟锛涘悓鏃讹紝鎴戜滑涔熻嚧鍔涗簬鍖栧鍝佺敤澶氳偨鐨勭爺鍙戜笌鐢熶骇銆侟/p>
閭:
鍏徃鍦板潃:
娴欐睙鐪佸寲瀛﹀師鏂欒嵂鍩哄湴涓存捣鍥尯涓滄捣绗洓澶ч亾5鍙